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OPK-88004

Aliases: OPK88004

Last verified: 2026-09-23

Clinical trialsModerate evidenceSARMsLow interest

The short version

A SARM with a unique profile: increases bone mass without enlarging the prostate — studied for osteoporosis and (paradoxically) BPH. Status: in clinical trials. Not approved; WADA-banned (S1).

Identity & type

Molecular type
SARM
Origin
A SARM with a unique profile: increases bone mass without enlarging the prostate — studied for osteoporosis and (paradoxically) BPH.

Mechanism of action

Tissue-selective AR modulation; antiproliferative on prostate preclinically.

Dosing & routes

Official / clinical context

No approved official document exists for OPK-88004. Any protocols mentioned are to be read as information, not as a recommendation.

Regulator-approved labeling and published study designs — never a recommendation.

Community-reported practice

Trials: 5–25 mg/day. No meaningful community experiences; trials show bone-density gains.

Unverified self-reports. Not medical advice. Not endorsement.

Expected effects (community)

No meaningful community experiences; trials show bone-density gains.

Protocol — official vs community

Official / label

No official protocol exists — this compound has no approved product.

Community (anecdotal)

Structured protocol data for this entry is coming.

Human evidence

Phase II (OPKO Health): bone mineral density in men.

Preclinical evidence

Preclinical literature preceded the clinical trials; details vary by compound.

Known risks

  • Mild GI upset, fatigue.characterized
  • WADA prohibition (S1 anabolic agents)characterized

Teal: characterized in clinical/labeling contexts. Amber: theoretical or reported outside controlled settings.

Unknowns & evidence gaps

  • Long-term safety in off-label use

Frequently asked questions

References

Systematic references are being expanded; verify sources directly before any decision.